Biotin-guided anticancer drug delivery with acidity-triggered drug release.

نویسندگان

  • Soyeon Park
  • Eunjin Kim
  • Won Young Kim
  • Chulhun Kang
  • Jong Seung Kim
چکیده

A novel biotin-guided anticancer drug delivery system, prodrug , consisting of biotin, nitrobenzene, and doxorubicin, with acid-triggered drug releasing capability was synthesized. Its cellular uptake and anticancer activity are selective to the HepG2 cell line over the WI-38 cell line, as revealed by fluorescence confocal microscopic experiments and MTT assay.

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عنوان ژورنال:
  • Chemical communications

دوره 51 45  شماره 

صفحات  -

تاریخ انتشار 2015